General Information of Binding Target of SBP (BTS) (ID: ST00114)
BTS Name
Apoptosis regulator Bcl-X
Synonyms
Bcl-2-like protein 1
BTS Type
Protein
Family
Bcl-2 family
Gene Name
bcl-xl
Organism
Felis catus (Cat) (Felis silvestris catus)
UniProt ID
Q8SQ42
UniProt Entry
Q8SQ42_FELCA
PFam
PF00452 ; PF02180
Gene ID
493701
Sequence
MSQSNRELVVDFLSYKLSQKGYSWSRFSDVEENRTEAPEGTESEMETPSAINGNPSWHLA
DSPAVNGATGHSSSLDAREVIPMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAY
QSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEP
WIQENGGWDTFVELYGNNAAAESRKGQERSNRWFLTGMTVAGVVLLGSLFSRK
Sequence Length
233
Synthetic Binding Protein (SBP) Targeting This BTS
SBP Name Highest Status Mechanism Affinity Application Details Ref
DARPin anti-Bcl-2/BCL-XL/Bcl-W 008_C6 Research Inhibitor Kd: 1.0 nM Cancers [ICD-11: 2D4Z]
SBP Info
[1]
References
1 From DARPins to LoopDARPins: novel LoopDARPin design allows the selection of low picomolar binders in a single round of ribosome display. J Mol Biol. 2014 Feb 6;426(3):691-721.